RPR-260243

SKU: orb1706687

Description

RPR-260243 is a novel small molecule that activates the HERG potassium channel. It can reverse the inhibition of HERG currents caused by dofetilide (IC50 = 58 nM), making it a valuable pharmacological tool for in vitro cardiac electrophysiology and arrhythmia research.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 668463-35-2
• MW: 510.5
• Formula: C₂₈H₂₅F₃N₂O₄
• SMILES: COc1ccc2nccc(C(=O)CC[C@@H]3CCN(CC#Cc4cc(F)cc(F)c4F)C[C@@H]3C(O)=O)c2c1
• Target: Potassium Channel,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

11466357