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Elagolix

SKU: orb3174300

Description

Elagolix is an orally active, highly effective, selective non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRH receptor) with a dissociation constant (KD) of 54 pM, as well as an NFAT inhibitor, and is utilized in researching endometriosis-related pain.

Research Area

Pharmacology & Drug Discovery

Images & Validation

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Key Properties

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CAS Number2323071-30-1
MW631.6
FormulaC32H30F5N3O5
SMILESO=C(O)CCCNC(C=1C=CC=CC1)CN2C(=O)C(C=3C=CC=C(OC)C3F)=C(N(C2=O)CC=4C(F)=CC=CC4C(F)(F)F)C
TargetGNRH Receptor

Storage & Handling

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Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Quality Guarantee

Quality Guarantee

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Protocol Information