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Pimethixene maleate
Catalog Number: orb1089596
| Catalog Number | orb1089596 |
|---|---|
| Category | Small Molecules |
| Description | Pimethixene (Pimetixene) maleate, an antihistamine, anntimigraine agent and antiserotonergic compound, is a highly potent antagonist of a broad range of monoamine receptors, including a variety of serotonin receptors. Pimethixene maleate inhibits 5-HT2A, 5-HT2B, 5-HT2C, 5-HT1A, 5-HT1B, 5-HT6, 5-HT7, Adrenergic α-1A, Dopamine D1 Receptor, Dopamine D2 Receptor, Dopamine D4.4 Receptor, Histamine H1 Receptor, Muscarinic M1 and Muscarinic M2 with pKi of 10.22, 10.44, 8.42, 7.63, < 5, 7.30, 7.28, 7.61, 6.37, 8.19, 7.54, 10.14, 8.61 and 9.38, respectively.,5-HT2B [1](Cell-free assay) 5-HT2A [1](Cell-free assay) Histamine H1 Receptor [1](Cell-free assay) Muscarinic M2 [1](Cell-free assay) Muscarinic M1 [1](Cell-free assay) View More 10.44(pKi) 10.22(pKi) 10.14(pKi) 9.38(pKi) 8.61(pKi) |
| CAS Number | [13187-06-9] |
| MW | 409.498025178909 |
| SMILES | OC(/C=C/C(=O)O)=O.CN1CC/C(=C2/C3=CC=CC=C3SC3=CC=CC=C/23)/CC1 |
| Formula | C23H23NO4S |
| Note | For research use only |
| Expiration Date | 12 months from date of receipt. |
Pimethixene maleate [orb1708846]
98%
13187-06-9
409.5
C23H23NO4S
25 mg, 10 mg, 50 mg, 5 mg, 1 ml x 10 mm (in DMSO)
