PF-05190457

• Catalog Number: orb2655950
• Category: Small Molecules
• Description: A potent, selective, and orally bioavailable ghrelin receptor (GHSR) inverse agonist with binding pKi of 8.36; displays excellent off-target activity in the CEREP panel at 10 uM with exception of serotonin 5-HT2B (IC50=3.7 uM).
• CAS Number: 1334782-79-4
• Purity: > 98% (HPLC)
• MW: 512.7
• Formula: C₂₉H₃₂N₆OS
• Target: GHSR
• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Note: For research use only
• Expiration Date: 12 months from date of receipt.