Orantinib (TSU-68)

SKU: orb146256

Description

SU6668 has greatest potency against PDGFR autophosphorylation with Ki of 8 nM, but also strongly inhibits Flk-1 and FGFR1 trans-phosphorylation, little activity against IGF-1R, Met, Src, Lck, Zap70, Abl and CDK2; does not inhibit EGFR.

Key Properties

• CAS Number: 252916-29-3
• MW: 482.53
• Purity: >98%
• Formula: C₂₈H₂₆N₄O₄
• SMILES: C(O)(=O)CCC1C(C)=C(/C=C2/C3=C(NC/2=O)C=CC=C3)NC=1C

Storage & Handling

• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only