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Orantinib (TSU-68)

SKU: orb146256

Description

SU6668 has greatest potency against PDGFR autophosphorylation with Ki of 8 nM, but also strongly inhibits Flk-1 and FGFR1 trans-phosphorylation, little activity against IGF-1R, Met, Src, Lck, Zap70, Abl and CDK2; does not inhibit EGFR.

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Key Properties

CAS Number252916-29-3
MW482.53
Purity>98%
FormulaC28H26N4O4
SMILESC(O)(=O)CCC1C(C)=C(/C=C2/C3=C(NC/2=O)C=CC=C3)NC=1C

Storage & Handling

Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Orantinib (TSU-68)

Chemical structure of Orantinib (TSU-68)

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Orantinib (TSU-68) (orb146256)

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100 mg
$ 460.00
250 mg
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1 g
$ 1,750.00
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