Ocaperidone

SKU: orb1304145

Description

Ocaperidone is a potent small molecule antagonist with very high affinity for the dopamine D2 receptor. It is a valuable research tool for investigating dopaminergic pathways in neuropharmacology and psychiatry, suitable for both in vitro binding assays and in vivo behavioral studies.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 129029-23-8
• MW: 420.48
• Purity: 99.33% (May vary between batches)
• Formula: C₂₄H₂₅FN₄O₂
• SMILES: Cc1cccn2c1nc(C)c(CCN1CCC(CC1)c1noc3cc(F)ccc13)c2=O
• Target: Dopamine Receptor,5-HT Receptor
• Solubility: DMSO:Slightly soluble

Bioactivity

• Target IC50:
  5-HT1A receptor:8.08 (pKi, h5-HT 1A)|5-HT1A receptor:7.6 (pEC50, h5-HT 1A)|5-HT2:0.14 nM(Ki)|H1:1.6 nM (Ki)|α2:5.4 nM (Ki)|D2:0.75 nM (Ki)|α1:0.46 nM (Ki)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

inhibit, Ocaperidona, Ocaperidone, Inhibitor, Dopamine, Dopamine Receptor, DopamineReceptor, D2, 5-hydroxytryptamine Receptor, 5HTReceptor, 5-HT2, 5-HT Receptor, 5HT Receptor, Serotonin Receptor, R79598, R-79598, R 79598

Compound Identifiers

PubChem CID

71351