EPZ005687

• Catalog Number: orb180981
• Category: Small Molecules
• Description: EPZ-005687 is a potent and selective inhibitor of EZH2 with Ki of 24 nM, 50-fold selectivity against EZH1 and 500-fold selectivity against 15 other protein methyltransferases.
• CAS Number: [1396772-26-1]
• MW: 539.6679
• SMILES: O1C([H])([H])C([H])([H])N(C([H])([H])C1([H])[H])C([H])([H])C1C([H])=C([H])C(=C([H])C=1[H])C1=C([H])C(C(N([H])C([H])([H])C2C(N([H])C(C([H])([H])[H])=C([H])C=2C([H])([H])[H])=O)=O)=C2C([H])=NN(C2=C1[H])C1([H])C([H])([H])C([H])([H])C([H])([H])C1([H])[H]
• Formula: C₃₂H₃₇N₅O₃
• Note: For research use only
• Expiration Date: 12 months from date of receipt.

Chemical structure of EPZ005687.