Enrasentan edamine

• Catalog Number: orb2815709
• Category: Small Molecules
• Description: Enrasentan (also known as SB-217242) is a dual receptor endothelin antagonist with a higher affinity for the ET(A) receptor. In animal models of hypertension and cardiac hypertrophy, this compound reduces blood pressure, prevents cardiac hypertrophy, and preserves myocardial function. Enrasentan enhances survival rates, limits left ventricular remodeling, and maintains myocardial performance in hypertensive cardiac hypertrophy and dysfunction.
• CAS Number: 183507-63-3
• MW: 536.60
• SMILES: NCCN.OC([C@H]1[C@H](C2=C(C=C(C=C2)OC)OCCO)C3=CC(OCCC)=CC=C3[C@@H]1C4=CC=C(OCO5)C5=C4)=O.OC([C@H]6[C@H](C7=C(C=C(C=C7)OC)OCCO)C8=CC(OCCC)=CC=C8[C@@H]6C9=CC=C(OCO%10)C%10=C9)=O
• Formula: C₃₀H₃₄NO₈
• Storage: -20°C
• Note: For research use only
• Expiration Date: 12 months from date of receipt.