Eletriptan hydrobromide

SKU: orb1225914

Description

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist; significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease; displays antimigraine activity.Migrainev Approved.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 177834-92-3
• MW: 463.43
• Purity: >98% (HPLC)
• Formula: C₂₂H₂₆N₂O₂S.HBr
• SMILES: CN1CCC[C@@H]1CC2=CNC3=C2C=C(C=C3)CCS(=O)(=O)C4=CC=CC=C4.Br
• Target: 5-HT Receptor
• Solubility: DMSO: 46.3 mg/mL (100 mM) （ < 1 mg/ml refers to the product slightly soluble or insoluble )

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

UK 116044 hydrobromide

Quick Database Links

Gene Symbol

5-HT Receptor