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DPCPX

SKU: orb1305827

Description

DPCPX

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number102146-07-6
MW304.39
Purity99.93% (May vary between batches)
FormulaC16H24N4O2
SMILESC(CC)N1C2=C(NC(=N2)C3CCCC3)C(=O)N(CCC)C1=O
TargetAdenosine Receptor
SolubilityEthanol:< 1 mg/mL (insoluble or slightly soluble);DMSO:3.05 mg/mL (10.02 mM)

Bioactivity

Target IC50
[3H]-NECA binding to A2 receptor (rat striatal membranes):340 nM (Ki)|[3H]-CHA binding to A1 receptor (rat whole brain membranes):0.46 nM (Ki)
In Vivo
DPCPX, a selective adenosine A1 receptor antagonist, enhances the antidepressant-like effects of imipramine, escitalopram, and reboxetine in mice behavioral tests

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

AdenosineReceptor, Adenosine Receptor, A1, DPCPX, inhibit, Inhibitor, PD 116948, PD116948, PD-116948, P1 receptor

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Quality Guarantee

Quality Guarantee

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Key Properties

No computed properties available.

Protocol Information

Available Sizes

Select a size below

5 mg
$ 80.00
10 mg
$ 90.00
1 ml x 10 mM (in DMSO)
$ 90.00
25 mg
$ 110.00
50 mg
$ 140.00
DispatchUsually dispatched within 5-10 working days
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