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Dersimelagon

Dersimelagon

Catalog Number: orb1089631

DispatchUsually dispatched within 5-10 working days
$ 820.00
Catalog Numberorb1089631
CategorySmall Molecules
DescriptionDersimelagon, also known as MT-7117 and WHO 10832, is a novel, orally-administered, small molecule, selective melanocortin-1 receptor (MC1R) agonist that increases skin melanin without sun exposure and is being developed to increase light tolerance in EPP/XLP patients. Dersimelagon significantly boosted sunlight tolerance in patients with erythropoietic protoporphyria in a multicenter, phase 2, randomized trial.
CAS Number[1835256-48-8]
MW675.753224134445
SMILESF[C@]1(C(N2C[C@@H](COC)[C@H](C3=CC=C(C(F)(F)F)C=C3N3CCC(C(=O)O)CC3)C2)=O)CN(C[C@@H]1C1C=CC(=CC=1)OC)C1CCCC1
FormulaC36H45F4N3O5
NoteFor research use only
Expiration Date12 months from date of receipt.
  • Dersimelagon phosphate [orb1739873]

    0.98

    2490660-87-0

    773.75

    C36H48F4N3O9P

    25 mg, 100 mg, 50 mg
  • Dersimelagon [orb1702360]

    97.35%

    1835256-48-8

    675.75

    C36H45F4N3O5

    5 mg, 10 mg, 25 mg, 50 mg, 1 mg, 1 ml x 10 mm (in DMSO)