Degarelix (acetate)

SKU: orb525674

Description

Degarelix is a synthetic gonadotropin-releasing hormone receptor (GNRHR) antagonist (IC50 = 3 nM in HEK293 cells expressing the human receptor).

Key Properties

• CAS Number: 214766-78-6
• MW: 1692.33
• Formula: C₈₂H₁₀₃CLN₁₈O₁₆.C₂H₄O₂
• SMILES: CC(C)NCCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC1=CC=C(NC(N)=O)C=C1)NC(=O)[C@H](CC2=CC=C(C=C2)NC(=O)[C@@H]3NC(=O)NC(=O)C3)NC(=O)[C@H](CO)NC(=O)[C@@H](CC4C=NC=CC=4)NC(=O)[C@@H](CC5=CC=C(Cl)C=C5)NC(=O)[C@H](NC(C)=O)CC6C=C7C(C=CC=C7)=CC=6)C(=O)N8[C@H](CCC8

Storage & Handling

• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only