CPI-169 (racemate)

• Catalog Number: orb320151
• Category: Small Molecules
• Description: CPI-169 racemate is the racemate form of CPI-169, which is a novel and potent EZH2 inhibitor with IC50 < 1 nM(inhibition of the catalytic activity of PRC2); decreases cellular levels of H3K27me3 with an EC50 of 70 nM, and triggers cell cycle arrest and apo
• CAS Number: [1450655-76-1]
• MW: 528.664
• SMILES: O=C(C1=C(C)N(C(C2CCN(S(=O)(CC)=O)CC2)C)C3=C1C=CC=C3)NCC4=C(OC)C=C(C)NC4=O
• Formula: C₂₇H₃₆N₄O₅S
• Note: For research use only
• Expiration Date: 12 months from date of receipt.

Chemical structure of CPI-169 (racemate)