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CGRP antagonist 1

CGRP antagonist 1

Catalog Number: orb1708126

DispatchUsually dispatched within 3-5 working days
$ 450.00
Catalog Numberorb1708126
CategorySmall Molecules
DescriptionCGRP antagonist 1
CAS Number1123757-49-2
Purity98%
MW494.54
SMILESO=C1[C@]2(C=3C(N1)=NC=CC3)CC=4C(C2)=CC=C(NC(CN5C=6C(C7(C5=O)CCOCC7)=CC=CC6)=O)C4
FormulaC29H26N4O4
Biological ActivityCGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.
Storage-20°C
NoteFor research use only
Expiration Date12 months from date of receipt.
  • CGRP (8-37) (human) [orb1140506]

    > 95% by hplc

    3125.64 Da

    H-Val-Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Ser-Arg-Ser-Gly-Gly-Val-Val-Lys-Asn-Asn-Phe-Val-Pro-Thr-Asn-Val-Gly-Ser-Lys-Ala-Phe-NH2

    1 mg
  • MK-3207 [orb2664844]

    98.00%

    957118-49-9

    557.59

    C31H29F2N5O3

    25 mg, 5 mg, 1 mg, 50 mg, 10 mg
  • AC 187 TFA [orb1981522]

    98.00%

    3004.27

    C129H206F3N37O42

    50 mg, 5 mg
  • CALCB Protein, Human, Recombinant (mFc) [orb1955760]

    98.00%

    36.2 kDa (predicted); 37 kDa (reducing conditions)

    100 μg
  • BMS-927711(Rimegepant) [orb573258]

    [1289023-67-1]

    534.57

    C28H28F2N6O3

    250 mg, 1 g, 100 mg, 1 ml x 10 mm (in DMSO)