CERC-501 (LY-2456302)

• Catalog Number: orb385565
• Category: Small Molecules
• Description: CERC-501(LY-2456302) is a potent, selective antagonist of the kappa opioid receptor (KOR) (Ki = 0.81 nM vs. 24.0 nM and 155 nM for the μ-opioid receptor (MOR) and δ-opioid receptor (DOR), respectively.
• CAS Number: [1174130-61-0]
• MW: 418.50318
• SMILES: O=C(N)C1=CC=C(OC2=CC=C(CN3[C@H](C4=CC(C)=CC(C)=C4)CCC3)C=C2)C(F)=C1
• Formula: C₂₆H₂₇N₂O₂F
• Note: For research use only
• Expiration Date: 12 months from date of receipt.