AM 281

• Catalog Number: orb181102
• Category: Small Molecules
• Description: Potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively). Increases locomotor activity following systemic administration in vivo. Analog of SR141716A (Ki = 14 nM).
• CAS Number: [202463-68-1]
• MW: 557.21
• SMILES: O=C(C1=NN(C2=CC=C(Cl)C=C2Cl)C(C3=CC=C(I)C=C3)=C1C)NN4CCOCC4
• Formula: C₂₁H₁₉Cl₂IN₄O₂
• Note: For research use only
• Expiration Date: 12 months from date of receipt.

Chemical structure of AM 281