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Adenosine receptor antagonist 5

Adenosine receptor antagonist 5

Catalog Number: orb2664033

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Catalog Numberorb2664033
CategorySmall Molecules
DescriptionAdenosine receptor antagonist5 (Compound 39) serves as a selective antagonist for the human adenosine A3 receptor (hA3R) with a Ki of 12 nM. This compound inhibits the accumulation of IB-MECA-induced cAMP in NCI-H1792 cells and suppresses the proliferation of LK-2 and NCI-H1792 cancer cells. Additionally, Adenosine receptor antagonist5 exhibits a rapid metabolism rate in human liver microsomes.
Purity98.00%
Storage-20°C
NoteFor research use only
Expiration Date12 months from date of receipt.
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