Salvinorin A Carbamate

SKU: orb2282967

Description

Salvinorin A carbamate, a potent κ-opioid receptor (KOR) full agonist, exhibits nearly the same potency as salvinorin A, with EC50 values of 6.2 and 4.5 nM, respectively, for activating the human KOR to augment the binding of [35S]GTPγS. Enhancing biological stability, the addition of a carbamate group to salvinorin A reduces deacetylation.

Key Properties

• CAS Number: 858345-57-0
• MW: 433.457
• Formula: C₂₂H₂₇NO₈
• SMILES: COC(=O)[C@@H]1C[C@H](OC(N)=O)C(=O)[C@H]2[C@@]1(C)CC[C@H]1C(=O)O[C@@H](C[C@]21C)c1ccoc1
• Target: Others

Storage & Handling

• Storage: -20°C
• Disclaimer: For research use only

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