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Ac-RYYRIK-NH2 TFA

SKU: orb1981549

Description

Ac-RYYRIK-NH2 TFA acts as both a potent partial agonist for ORL1 when transfected in CHO cells (K d = 1.5 nM) and an endogenous ligand of ORL1. Moreover, it serves as a specific antagonist that inhibits G protein activation and competitively blocks the stimulation of [35S]-GTPγS binding to G proteins by nociceptin/orphanin FQ (noc/OFQ) in rat brain membranes and sections.

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Key Properties

MW1053.13
FormulaC46H71F3N14O11
TargetOpioid Receptor

Storage & Handling

Storage-20°C
DisclaimerFor research use only
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Ac-RYYRIK-NH2 TFA (orb1981549)

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(Recommended: An additional animal making an allowance for loss during the experiment)

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