K-(D-1-Nal)-FwLL-NH2 TFA

• Catalog Number: orb1981509
• Category: Small Molecules
• Description: K-(D-1-Nal)-FwLL-NH2 TFA is a potent, high-affinity inverse agonist of the ghrelin receptor with Ki values of 4.9 nM in COS7 cells and 31 nM in HEK293T cells, effectively inhibiting ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
• Purity: 98.00%
• MW: 1016.16
• Biological Activity: K-(D-1-Nal)-FwLL-NH2 TFA is a potent and high-affinity inverse agonist of the ghrelin receptor, exhibiting Ki values of 4.9 nM in COS7 cells and 31 nM in HEK293T cells. This compound effectively inhibits ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
• Formula: C₅₃H₆₈F₃N₉O₈
• Storage: -20°C
• Note: For research use only