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ARV-825

ARV-825

Catalog Number: orb1301793

DispatchUsually dispatched within 3-5 working days
$ 160.00
Catalog Numberorb1301793
CategorySmall Molecules
DescriptionARV-825
Purity97.54%
MW923.43
Biological ActivityARV-825, a heterobifunctional PROTAC (Proteolysis Targeting Chimera) that recruits BRD4 to the E3 ubiquitin ligase cereblon leading to fast, efficient, and prolonged degradation of BRD4 in all BL cell lines tested.
CAS Number[1818885-28-7]
FormulaC46H47ClN8O9S
SMILESCC=1C2=C(N3C([C@H](CC(NC4=CC=C(OCCOCCOCCOCCNC5=C6C(C(=O)N(C6=O)C7C(=O)NC(=O)CC7)=CC=C5)C=C4)=O)N=C2C8=CC=C(Cl)C=C8)=NN=C3C)SC1C
Storage-20°C
NoteFor research use only
  • ARV-825 [orb1225875]

    > 98% (HPLC)

    1818885-28-7

    923.4

    C46H47ClN8O9S

    1 g, 500 mg, 200 mg, 100 mg, 5 mg, 10 mg, 25 mg, 50 mg
  • ARV-825 [orb573167]

    306.33

    C19H15FN2O

    1 g, 100 mg, 250 mg, 1 ml x 10 mM (in DMSO)